SCHEMBL808060

SCHEMBL808060

c1ccc(-c2ccc3c(c2)C2(c4cc(-c5ccccc5)ccc4-3)c3cc(-c4ccccc4)ccc3-c3ccc(N4c5ccccc5Oc5ccccc54)cc32)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 7/20 0.38
PDE6D O43924 1/20 0.33
TDP2 O95551 1/20 0.33
FAAH O00519 2/20 0.33
MGLL Q99685 2/20 0.33
HTT P42858 2/20 0.33
ATM Q13315 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HSP90AA1 P07900 1/20 0.33
PKM P14618 1/20 0.33
P2RX4 Q99571 2/20 0.32
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
MEN1 O00255 1/20 0.31
APAF1 O14727 1/20 0.31
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
XBP1 P17861 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15183639 0.96 PDK2 (0.41) PDK2PDE6DHTTATMMEN1
SCHEMBL14823503 0.90 P2RX4 (0.36) PDK2P2RX4MAPTSMN1; SMN2NPSR1
SCHEMBL24647359 0.89 PDK2 (0.38) PDK2PDE6D
SCHEMBL18542241 0.88 PDK2 (0.38) PDK2PDE6DTDP2FAAHMGLL
SCHEMBL15030821 0.87 PDK2 (0.39) PDK2HTTATMMEN1APAF1
SCHEMBL15183677 0.87 PDK2 (0.40) PDK2PDE6DTDP2FAAHMGLL
SCHEMBL808007 0.86 PDK2 (0.39) PDK2PDE6DTDP2FAAHMGLL
SCHEMBL807996 0.85 PDK2 (0.35) PDK2HTTP2RX4MEN1LMNA
SCHEMBL21867888 0.85 PDK2 (0.36) PDK2PDE6DFAAHMGLLHTT
SCHEMBL14550933 0.85 PDK2 (0.31) PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2826079-B1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2021-01-20 EP disclosed
US-10454040-B2 Materials for electronic devices MERCK PATENT GMBH (DE) 2019-10-22 US disclosed
US-10270052-B2 Electronic device MERCK PATENT GMBH (DE) 2019-04-23 US disclosed
EP-3460864-A1 ELECTRONIC DEVICES Merck Patent GmbH (DE) 2019-03-27 EP disclosed
US-20180138439-A1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2018-05-17 US disclosed
US-20180138439-A1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2018-05-17 US disclosed
US-9947874-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2018-04-17 US disclosed
US-9947874-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2018-04-17 US disclosed
EP-2907173-B1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2018-03-21 EP disclosed
US-9917272-B2 Electronic device MERCK PATENT GMBH (DE) 2018-03-13 US disclosed
US-20150236261-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-08-20 US disclosed
US-20150236261-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-08-20 US disclosed
US-20150115239-A1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-04-30 US disclosed
US-20150115239-A1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-04-30 US disclosed
EP-2616428-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2014-12-24 EP disclosed
WO-2014044344-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2014-03-27 WO disclosed
WO-2013135352-A1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2013-09-19 WO disclosed
US-20130207046-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2013-08-15 US disclosed
US-20130207046-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2013-08-15 US disclosed
WO-2012034627-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2012-03-22 WO disclosed