SCHEMBL8081390

SCHEMBL8081390

CC(=O)Nc1cn2c3c(cccc13)CCC2

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.59
MTNR1B P49286 7/20 0.59
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HSD17B10 Q99714 2/20 0.44
MCL1 Q07820 1/20 0.44
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
OPA1 O60313 1/20 0.42
EIF5B O60841 1/20 0.42
MET P08581 1/20 0.42
HMOX2 P30519 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2260100 0.84 MTNR1A (0.49) MTNR1AMTNR1BHTR2AHTR2CHSD17B10
SCHEMBL13087729 0.79 MTNR1A (0.50) MTNR1AMTNR1BHTR2AHTR2CHSD17B10
SCHEMBL2020434 0.79 MTNR1A (0.59) MTNR1AMTNR1BHTR2AHTR2CHSD17B10
SCHEMBL2024854 0.78 MTNR1A (0.56) MTNR1AMTNR1BHTR2AHTR2CHSD17B10
SCHEMBL10100276 0.75 HTR2A (0.59) MTNR1AMTNR1BHTR2AHTR2CHSD17B10
SCHEMBL1395799 0.74 HTR2A (0.52) MTNR1AMTNR1BHTR2AHTR2CHSD17B10
SCHEMBL1395855 0.74 HTR2A (0.55) MTNR1AMTNR1BHTR2AHTR2CHSD17B10
SCHEMBL1719811 0.74 MTNR1A (0.51) MTNR1AMTNR1BHTR2AHTR2CHSD17B10
SCHEMBL3065255 0.74 MTNR1A (0.53) MTNR1AMTNR1B
SCHEMBL3060070 0.74 MTNR1A (0.53) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026446-A9 HDAC INHIBITORS ARQULE, INC. (US) 2010-03-11 WO disclosed
WO-2009026446-A2 HDAC INHIBITORS ARQULE, INC. (US) 2009-02-26 WO disclosed
CN-1312154-C Purine derivatives as kinase inhibitors LILLY CO ELI (US) 2007-04-25 CN disclosed
CN-1639165-A Purine derivatives as kinase inhibitors LILLY CO ELI (US) 2005-07-13 CN disclosed