SCHEMBL8081759

SCHEMBL8081759

CC1(C)CCOc2ccc(SI)cc21

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.45
RARG P13631 5/20 0.45
RARA P10276 4/20 0.45
RXRA P19793 3/20 0.43
CYP26A1 O43174 1/20 0.40
CYP26B1 Q9NR63 1/20 0.40
AKR1B1 P15121 1/20 0.35
HNF4A P41235 1/20 0.35
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
MAP3K14 Q99558 1/20 0.33
SSTR5 P35346 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4373360 0.84 RARB (0.45) RARBRARGRARARXRACYP26A1
SCHEMBL9188117 0.84 RARB (0.48) RARBRARGRARARXRACYP26A1
SCHEMBL4370337 0.81 RARB (0.43) RARBRARGRARARXRACYP26A1
SCHEMBL3456678 0.79 RARB (0.51) RARBRARGRARARXRACYP26A1
SCHEMBL10557225 0.79 RARB (0.44) RARBRARGRARARXRACYP26A1
SCHEMBL9190581 0.79 RARB (0.53) RARBRARGRARARXRACYP26A1
SCHEMBL8293244 0.76 RARA (0.49) RARBRARGRARARXRACYP26A1
SCHEMBL18211725 0.76 MAP3K14 (0.50) RARBRARGRARARXRACYP26A1
SCHEMBL2599701 0.75 RARA (0.48) RARBRARGRARARXRACYP26A1
SCHEMBL9053722 0.75 RARA (0.48) RARBRARGRARARXRACYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0740665-B1 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES ALLERGAN SALES INC (US) 2000-12-06 EP disclosed
EP-0740665-A1 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES Allergan (US) 1996-11-06 EP disclosed
US-5519150-A Process for preparing 4,4-dialkyl-6-halo-chromans or thiochromans useful as pharmaceutical intermediates ALLERGAN (US) 1996-05-21 US disclosed
WO-1995019973-A2 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES ALLERGAN (US) 1995-07-27 WO disclosed
US-5420295-A Process for preparing 4,4-dialkyl-6-halo-chromans or thiochromans useful as pharmaceutical intermediates ALLERGAN, INC. (US) 1995-05-30 US disclosed