SCHEMBL8081871

SCHEMBL8081871

C=CCN1C[C@@H](C)N(C(c2cccc(O)c2)c2ccccc2C#N)CC1C

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
HPGD P15428 1/20 0.58
OPRM1 P35372 1/20 0.58
OPRK1 P41145 1/20 0.58
SIGMAR1 Q99720 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6932686 1.00 OPRD1 (0.58) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL8030090 0.87 CYP1A2 (0.45) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6653135 0.87 CYP1A2 (0.45) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL15080469 0.86 OPRD1 (0.61) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6465443 0.86 OPRD1 (0.61) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6465439 0.86 OPRD1 (0.61) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6936322 0.86 OPRD1 (0.61) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6936320 0.86 OPRD1 (0.61) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6659217 0.86
SCHEMBL8081874 0.85 OPRD1 (0.63) OPRD1CYP1A2CYP3A4CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711289-B1 PIPERAZINE COMPOUNDS USED IN THERAPY DELTA PHARMACEUTICALS INC (US) 2000-08-23 EP disclosed