SCHEMBL8082610

SCHEMBL8082610

CNCCc1cccc2ccoc12

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.48
HTR2C P28335 1/20 0.48
TAAR1 Q96RJ0 4/20 0.44
EED O75530 1/20 0.40
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
ATM Q13315 1/20 0.37
KCNH2 Q12809 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR1A P08908 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31137328 0.82 HTR2A (0.47) HTR2AHTR2CEEDKCNH2
SCHEMBL3794977 0.80 EED (0.43) HTR2AHTR2CEEDKCNH2
SCHEMBL3793855 0.77 EED (0.41) HTR2AHTR2CEEDKCNH2
SCHEMBL34462948 0.77 EED (0.43) HTR2AHTR2CTAAR1EEDKCNH2
SCHEMBL28181295 0.77 EED (0.43) HTR2AHTR2CEEDKCNH2
SCHEMBL2610674 0.76 GABRA1 (0.46) HTR2AHTR2CEEDKCNH2
SCHEMBL2094027 0.74 EED (0.41) HTR2AHTR2CEEDKCNH2
SCHEMBL20354322 0.73 GABRA1 (0.48) HTR2AHTR2CEEDKCNH2
SCHEMBL24336535 0.72 EED (0.43) HTR2AHTR2CEEDKCNH2KDM4E
SCHEMBL5541627 0.72 EED (0.40) HTR2AHTR2CEEDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6063810-A ENANTIOMORPHS SYNTHELABO (FR) 2000-05-16 US disclosed
EP-0688320-B1 TRICYCLIC BENZODIAZEPINS, THEIR USE AND PREPARATION NOVO NORDISK AS (DK) 1999-05-06 EP disclosed
US-5512562-A FOR CENTRAL NERVOUS SYSTEM DISORDERS; PSYCHOSIS, DEPRESSION, SLEEP DISORDERS, PARKINSON*S DISEASE, STROKE NOVO NORDISK A/S (DK) 1996-04-30 US disclosed
EP-0688320-A1 TRICYCLIC BENZODIAZEPINS, THEIR USE AND PREPARATION NOVO NORDISK A/S (DK) 1995-12-27 EP disclosed
WO-1994020472-A1 HETEROCYCLIC COMPOUNDS, THEIR USE AND PREPARATION NOVO NORDISK A/S (DK) 1994-09-15 WO disclosed