SCHEMBL8083231

SCHEMBL8083231

CC=CC=CCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.49
ALDH1A1 P00352 2/20 0.43
CA12 O43570 2/20 0.43
CA9 Q16790 2/20 0.43
CA2 P00918 1/20 0.43
GLS O94925 1/20 0.42
DRD3 P35462 1/20 0.41
RPS6KA2 Q15349 1/20 0.40
ALDH3A1 P30838 1/20 0.40
RCE1 Q9Y256 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083226 1.00 CASP3 (0.49) CASP3ALDH1A1CA12CA9CA2
SCHEMBL12223397 0.87 CA12 (0.54) CASP3ALDH1A1CA12CA9CA2
SCHEMBL10237149 0.87 CA12 (0.54) CASP3ALDH1A1CA12CA9CA2
SCHEMBL6010522 0.87 CA12 (0.54) CASP3ALDH1A1CA12CA9CA2
SCHEMBL4468251 0.82 CASP3 (0.60) CASP3ALDH1A1CA12CA9GLS
SCHEMBL8950475 0.82 CASP3 (0.60) CASP3ALDH1A1CA12CA9GLS
SCHEMBL4476083 0.82 CASP3 (0.60) CASP3ALDH1A1CA12CA9GLS
SCHEMBL8091163 0.80 CASP3 (0.59) CASP3ALDH1A1CA12CA9GLS
SCHEMBL7185886 0.80 CASP3 (0.59) CASP3ALDH1A1CA12CA9GLS
SCHEMBL5394867 0.79 CASP3 (0.56) CASP3ALDH1A1CA12CA9GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0682030-B1 8-Amino-10(azabicycloalkyl)-pyrido[1,2,3-d,e] [1,3,4] benzoxadiazine derivatives, process for their preparation and antibacterial agents containing them BAYER AG (DE) 2000-07-05 EP disclosed
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed
EP-0647644-B1 Antibacterial pyrido 1,2,3-d,e 1,3,4 benzoxacin derivatives BAYER AG (DE) 1997-11-05 EP disclosed
US-5556979-A ANIMAL FEEDS BAYER AKTIENGESELLSCHAFT (DE) 1996-09-17 US disclosed
EP-0588166-B1 Antibacterial 7-isoindolinyl-quinolone and naphthyridone derivatives BAYER AG (DE) 1996-06-05 EP disclosed
EP-0682030-A1 8-Amino-10(azabicycloalkyl)-pyrido[1,2,3-d,e] [1,3,4] benzoxadiazine derivatives, process for their preparation and antibacterial agents containing them BAYER AG (DE) 1995-11-15 EP disclosed
EP-0647644-A1 Antibacterial pyrido 1,2,3-d,e 1,3,4 benzoxacin derivatives BAYER AG (DE) 1995-04-12 EP disclosed
EP-0588166-A2 Antibacterial 7-isoindolinyl-quinolone and naphthyridone derivatives BAYER AG (DE) 1994-03-23 EP disclosed