SCHEMBL808393

SCHEMBL808393

CC1(C)c2ccccc2N(c2cccc(-c3ccccc3)c2)c2ccc(-c3ccc4c(c3)C3(c5ccccc5-c5ccccc53)c3ccccc3-4)cc21

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 13/20 0.39
FAAH O00519 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HSP90AA1 P07900 1/20 0.37
PKM P14618 1/20 0.37
HTT P42858 1/20 0.37
ATM Q13315 1/20 0.37
MGLL Q99685 1/20 0.37
PGR P06401 4/20 0.35
PDE6D O43924 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807997 0.94 PDK2 (0.39) PDK2PGRPDE6D
SCHEMBL19530841 0.93 PDK2 (0.39) PDK2HTTATMPGRPDE6D
SCHEMBL15183560 0.93 PDK2 (0.40) PDK2FAAHMGLLPGRPDE6D
SCHEMBL15183561 0.93 PDK2 (0.40) PDK2FAAHMGLLPGRPDE6D
SCHEMBL10038900 0.93 PDK2 (0.42) PDK2ALDH1A1HTTATMPGR
SCHEMBL808313 0.93 PGR (0.40) PDK2ALDH1A1PGR
SCHEMBL15183539 0.91 PDK2 (0.41) PDK2HTTATMPGR
SCHEMBL15183644 0.91 PDK2 (0.41) PDK2HTTATMPGRPDE6D
SCHEMBL15183557 0.90 PDK2 (0.42) PDK2FAAHMGLLPGRPDE6D
SCHEMBL15290070 0.90 PDK2 (0.42) PDK2FAAHMGLLPGRPDE6D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2826079-B1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2021-01-20 EP disclosed
US-10454040-B2 Materials for electronic devices MERCK PATENT GMBH (DE) 2019-10-22 US disclosed
US-10270052-B2 Electronic device MERCK PATENT GMBH (DE) 2019-04-23 US disclosed
EP-3460864-A1 ELECTRONIC DEVICES Merck Patent GmbH (DE) 2019-03-27 EP disclosed
US-20180138439-A1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2018-05-17 US disclosed
US-20180138439-A1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2018-05-17 US disclosed
US-9947874-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2018-04-17 US disclosed
US-9947874-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2018-04-17 US disclosed
EP-2907173-B1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2018-03-21 EP disclosed
US-9917272-B2 Electronic device MERCK PATENT GMBH (DE) 2018-03-13 US disclosed
US-20150270506-A1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2015-09-24 US disclosed
US-20150236261-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-08-20 US disclosed
US-20150236261-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-08-20 US disclosed
US-20150115239-A1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-04-30 US disclosed
US-20150115239-A1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-04-30 US disclosed
EP-2616428-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2014-12-24 EP disclosed
WO-2013135352-A1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2013-09-19 WO disclosed
US-20130207046-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2013-08-15 US disclosed
US-20130207046-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2013-08-15 US disclosed
WO-2012034627-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2012-03-22 WO disclosed