SCHEMBL8084448

SCHEMBL8084448

COc1ccc([C@H]2CC[C@H]3[C@@H]4[C@@H](C)C[C@H]5NC(=O)CC[C@]5(C)[C@H]4CC[C@]23C)cc1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 6/20 0.52
SRD5A1 P18405 5/20 0.52
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
AR P10275 1/20 0.37
SHBG P04278 1/20 0.37
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084449 1.00 SRD5A2 (0.52) SRD5A2SRD5A1DDB1CRBNAR
SCHEMBL8023123 0.85 SRD5A1 (0.53) SRD5A2SRD5A1AR
SCHEMBL8016811 0.83 SRD5A2 (0.49) SRD5A2SRD5A1AR
SCHEMBL8096297 0.82 SRD5A1 (0.55) SRD5A2SRD5A1
SCHEMBL8096293 0.82 SRD5A1 (0.55) SRD5A2SRD5A1
SCHEMBL8092620 0.79 SRD5A1 (0.52) SRD5A2SRD5A1
SCHEMBL8092618 0.79 SRD5A1 (0.52) SRD5A2SRD5A1
SCHEMBL8996777 0.78 SRD5A2 (0.52) SRD5A2SRD5A1ARSHBG
SCHEMBL8018780 0.78 SRD5A2 (0.47) SRD5A2SRD5A1AR
SCHEMBL8016817 0.78 SRD5A2 (0.43) SRD5A2SRD5A1ARSHBG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0756481-B1 17$g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO INC (US) 2000-12-27 EP disclosed
EP-0756481-A4 17-g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO INC (US) 1998-11-18 EP disclosed
EP-0756481-A1 17$g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO. INC. (US) 1997-02-05 EP disclosed
US-5525608-A ANTIACNE AGENT, SKIN DISORDERS, GLANDULAR DISORDERS MERCK & CO., INC. (US) 1996-06-11 US disclosed
WO-1995028928-A1 17β-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO., INC. (US) 1995-11-02 WO disclosed