SCHEMBL8996777

SCHEMBL8996777

Cc1ccc(OC2CC[C@H]3[C@@H]4C(C)CC5NC(=O)CC[C@]5(C)[C@@H]4CC[C@]23C)cc1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 8/20 0.52
SRD5A1 P18405 7/20 0.52
AR P10275 1/20 0.37
SHBG P04278 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL917575 0.83 SRD5A2 (0.45) SRD5A2SRD5A1ARSHBG
SCHEMBL8016670 0.79 SRD5A2 (0.55) SRD5A2SRD5A1ARSHBG
SCHEMBL8084449 0.78 SRD5A2 (0.52) SRD5A2SRD5A1ARSHBG
SCHEMBL8084448 0.78 SRD5A2 (0.52) SRD5A2SRD5A1ARSHBG
SCHEMBL7613727 0.77 SRD5A2 (0.51) SRD5A2SRD5A1AR
SCHEMBL7903652 0.77 SRD5A2 (0.48) SRD5A2SRD5A1ARSHBG
SCHEMBL7613719 0.77 SRD5A2 (0.51) SRD5A2SRD5A1AR
SCHEMBL3278549 0.76 SRD5A2 (0.61) SRD5A2SRD5A1AR
SCHEMBL3276274 0.76 SRD5A1 (0.52) SRD5A2SRD5A1AR
SCHEMBL8530143 0.75 SRD5A1 (0.47) SRD5A2SRD5A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724592-A1 16-SUBSTITUTED-4-AZA-ANDROSTANE 5-ALPHA-REDUCTASE ISOZYME 1 INHIBITORS MERCK & CO. INC. (US) 1996-08-07 EP disclosed
WO-1995011254-A1 16-SUBSTITUTED-4-AZA-ANDROSTANE 5-ALPHA-REDUCTASE ISOZYME 1 INHIBITORS MERCK & CO., INC. (US) 1995-04-27 WO disclosed