SCHEMBL8086000

SCHEMBL8086000

O=C(O)CN1CCCCC(NS(=O)(=O)Cc2ccccc2)C1=O

nearest known ligand 0.71

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
F2 P00734 14/20 0.71
PRSS1 P07477 9/20 0.67
F10 P00742 9/20 0.67
PRSS2 P07478 3/20 0.67
PRSS3 P35030 3/20 0.67
ACE P12821 6/20 0.60
MME P08473 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5860343 1.00 F2 (0.71) F2PRSS1F10PRSS2PRSS3
SCHEMBL10795369 0.77 ACE (0.80) ACEMME
SCHEMBL10795378 0.77 ACE (0.80) ACEMME
SCHEMBL6601810 0.77 CASP3 (0.68) ACEMME
SCHEMBL10792401 0.76 ACE (0.88) ACEMME
SCHEMBL10792409 0.76 ACE (0.88) ACEMME
SCHEMBL9058169 0.76 ACE (0.67) F2ACEMME
SCHEMBL8073897 0.76 ACE (0.67) F2ACEMME
SCHEMBL7347032 0.75 ACE (1.00) ACEMME
SCHEMBL7347023 0.75 ACE (1.00) ACEMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6034215-A 3-amino-2-oxo-1-piperidnercetic derivatives as enzyme inhibitors CORVAS INTERNATIONAL, INC. (US) 2000-03-07 US disclosed
US-5703208-A ANTICOAGULANTS CORVAS INTERNATIONAL, INC. (US) 1997-12-30 US disclosed
EP-0802923-A1 3-AMINO-2-OXO-1-PIPERIDINEACETIC DERIVATIVES AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1997-10-29 EP disclosed
WO-1995035311-A9 3-AMINO-2-OXO-1-PIPERIDINEACETIC DERIVATIVES AS ENZYME INHIBITORS 1996-02-01 WO disclosed
WO-1995035311-A1 3-AMINO-2-OXO-1-PIPERIDINEACETIC DERIVATIVES AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1995-12-28 WO disclosed