SCHEMBL8088945

SCHEMBL8088945

N#Cc1ccc(Cc2cncn2CCN)cc1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 16/20 0.55
CYP11B2 P19099 16/20 0.55
CYP19A1 P11511 1/20 0.50
HRH3 Q9Y5N1 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8390918 0.86 CYP11B1 (0.62) CYP11B1CYP11B2CYP19A1HRH3
SCHEMBL6180585 0.80 CYP11B1 (0.44) CYP11B1CYP11B2HRH3LOXL2
SCHEMBL5891862 0.79 CYP11B1 (0.55) CYP11B1CYP11B2CYP19A1
Hydrochloric Acid SCHEMBL8174417 0.78 CYP11B1 (0.54) CYP11B1CYP11B2CYP19A1
SCHEMBL8298245 0.78 CYP11B1 (0.56) CYP11B1CYP11B2CYP19A1
SCHEMBL8387542 0.77 CYP11B1 (0.46) CYP11B1CYP11B2CYP19A1
SCHEMBL8097809 0.77 CYP11B1 (0.46) CYP11B1CYP11B2CYP19A1
SCHEMBL7475351 0.77 CYP11B1 (0.71) CYP11B1CYP11B2CYP19A1
SCHEMBL7507201 0.77 CYP11B1 (0.74) CYP11B1CYP11B2CYP19A1
Hydrochloric Acid SCHEMBL7473109 0.76 CYP11B1 (0.70) CYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127366-A ANTICARCINOGENIC OR ANTITUMOR AGENTS MERCK & CO., INC. (US) 2000-10-03 US disclosed
US-5817678-A IMIDAZOLE-CONTAINING PIPERIDINE DERIVATIVES, PEPTIDEMIMETIC MERCK & CO., INC. (US) 1998-10-06 US disclosed