SCHEMBL8089402

SCHEMBL8089402

O=C1c2cccc([N+](=O)[O-])c2C(=O)N1CCc1ccc(O)cc1

nearest known ligand 0.73

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.73
CA2 P00918 3/20 0.73
CA9 Q16790 3/20 0.73
CA4 P22748 1/20 0.73
CA12 O43570 2/20 0.56
ATM Q13315 1/20 0.53
ACHE P22303 1/20 0.51
ALDH1A1 P00352 5/20 0.50
POLB P06746 1/20 0.48
TDP1 Q9NUW8 2/20 0.48
MAPT P10636 1/20 0.48
APEX1 P27695 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 1/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5782961 0.85 CA1 (0.70) CA1CA2CA9CA4CA12
SCHEMBL5783029 0.84 CA1 (0.69) CA1CA2CA9CA4CA12
SCHEMBL11306933 0.81 CA1 (0.60) CA1CA2CA9CA4CA12
SCHEMBL11314968 0.81 CA1 (0.63) CA1CA2CA9CA4CA12
SCHEMBL8085887 0.80 CA1 (0.50) CA1CA2CA9CA4CA12
SCHEMBL11307275 0.80 POLB (0.64) CA1CA2CA9CA4CA12
SCHEMBL28932673 0.79 CYP1B1 (0.50) CA1CA2CA9CA4CA12
SCHEMBL30956737 0.79 CYP1B1 (0.50) CA1CA2CA9CA4CA12
SCHEMBL8091427 0.79 CA1 (0.60) CA1CA2CA9CA4CA12
SCHEMBL4235928 0.78 ALDH1A1 (0.60) CA1CA2CA9CA4CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017919-A Compounds and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2000-01-25 US disclosed
EP-0887340-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL USE THEREOF Japan Tobacco Inc. (JP) 1998-12-30 EP disclosed