SCHEMBL8089497

SCHEMBL8089497

CC(C)(C)OC(=O)N1CCC(Oc2cc(F)c(C#N)cc2F)CC1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 13/20 0.56
PDE4D Q08499 3/20 0.47
PDE4A P27815 2/20 0.47
PDE4B Q07343 2/20 0.47
PDE4C Q08493 2/20 0.47
TBK1 Q9UHD2 2/20 0.46
KDM1A O60341 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088595 0.86 GPR119 (0.49) GPR119PDE4DPDE4APDE4BPDE4C
SCHEMBL18639877 0.85 SCN9A (0.53) GPR119
SCHEMBL4689209 0.83 GPR6 (0.40) GPR119
SCHEMBL223791 0.83 GPR119 (0.64) GPR119PDE4DPDE4APDE4BPDE4C
SCHEMBL3085652 0.83 GPR119 (0.55) GPR119PDE4DPDE4APDE4BPDE4C
SCHEMBL29964750 0.83 GPR119 (0.59) GPR119PDE4DPDE4APDE4BPDE4C
SCHEMBL30140081 0.82 GPR119 (0.47) GPR119PDE4BTBK1KDM1A
SCHEMBL31583681 0.82 GPR119 (0.54) GPR119
SCHEMBL29825828 0.81 GPR119 (0.47) GPR119TBK1
SCHEMBL1142588 0.81 GPR119 (0.53) GPR119PDE4DPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed