SCHEMBL8089616

SCHEMBL8089616

CC(C)(C)ON1CCC(Oc2ccc(CC(=O)N3CCC(N4C(=O)OCc5c(F)cccc54)CC3)c(OCC(F)(F)F)c2)CC1=C=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 20/20 0.61
AVPR2 P30518 7/20 0.61
AVPR1A P37288 7/20 0.61
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
CHRM4 P08173 1/20 0.39
HTR1A P08908 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR1E P28566 1/20 0.39
HTR1F P30939 1/20 0.39
HTR7 P34969 1/20 0.39
ADRA1A P35348 1/20 0.39
DRD3 P35462 1/20 0.39
HTR2B P41595 1/20 0.39
HTR3A P46098 1/20 0.39
HTR5A P47898 1/20 0.39
HTR6 P50406 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089362 0.88 OXTR (0.69) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8089437 0.84 OXTR (0.68) OXTRAVPR2AVPR1AHTR3EHTR3B
Hydrochloric Acid SCHEMBL8095229 0.83 OXTR (0.67) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8093360 0.82 OXTR (0.66) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8093364 0.80 OXTR (0.61) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8089301 0.78 OXTR (0.85) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL7333661 0.78 OXTR (0.42) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL8081394 0.77 OXTR (1.00) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL7333820 0.76 OXTR (0.41) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL8092986 0.75 OXTR (0.83) OXTRAVPR2AVPR1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed