SCHEMBL8090594

SCHEMBL8090594

CCCNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)O)CC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 8/20 0.40
KDR P35968 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NAMPT P43490 1/20 0.39
PIK3CA P42336 5/20 0.38
MTOR P42345 1/20 0.38
PIK3CG P48736 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
RAB9A P51151 1/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC3 O15379 1/20 0.37
MAPT P10636 1/20 0.37
KIT P10721 1/20 0.37
RXRA P19793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089827 0.91 PIK3CD (0.37) PIK3CDKDRPIK3CAMTORPIK3CG
SCHEMBL8081794 0.90 PIK3CA (0.44) NAMPTPIK3CAMTORPIK3CG
SCHEMBL8092884 0.87 KDR (0.41) PIK3CDKDRNAMPTPIK3CAKIT
SCHEMBL8098261 0.87 MTOR (0.43) PIK3CDMEN1KMT2APIK3CAMTOR
SCHEMBL8098056 0.86 KDM4E (0.38) PIK3CDKDRMEN1KMT2APIK3CA
SCHEMBL8095600 0.84 CA12 (0.39) PIK3CDMEN1KMT2ANAMPTHDAC1
SCHEMBL8088889 0.81 PIK3CD (0.44) PIK3CDKDRMEN1KMT2ANAMPT
SCHEMBL8099345 0.81 PIK3CD (0.44) PIK3CDKDRMEN1KMT2ANAMPT
SCHEMBL8083714 0.80 EPHX1 (0.45) KDRMEN1KMT2ACYP2C19RAB9A
SCHEMBL8096016 0.80 PIK3CD (0.43) PIK3CDKDRMEN1KMT2ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed