SCHEMBL8083714

SCHEMBL8083714

Nc1cc(C2(S(=O)O)CC2)nc(-c2ccc(NC(=O)NC3CCC3)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 9/20 0.45
RAB9A P51151 7/20 0.45
GAA P10253 1/20 0.45
KDR P35968 2/20 0.42
KIT P10721 1/20 0.42
FLT3 P36888 1/20 0.42
EPHX2 P34913 2/20 0.41
NPC1 O15118 7/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098261 0.85 MTOR (0.43) ALDH1A1MEN1KMT2A
SCHEMBL8095600 0.84 CA12 (0.39) EPHX2CA12CA1CA2CA9
SCHEMBL8099411 0.82 CA12 (0.44) EPHX1RAB9AGAAKDRKIT
SCHEMBL8089827 0.81 PIK3CD (0.37) KDR
SCHEMBL8099109 0.81 CA12 (0.43) EPHX1RAB9AGAAKDRKIT
SCHEMBL8090594 0.80 PIK3CD (0.40) RAB9AKDRKITCYP2C19MEN1
SCHEMBL8092884 0.80 KDR (0.41) KDRKITEPHX2
SCHEMBL8096200 0.79 EPHX1 (0.47) EPHX1RAB9AGAAKDRKIT
SCHEMBL8097694 0.79 CYP3A4 (0.42) EPHX1RAB9AGAAKDRKIT
SCHEMBL8092878 0.79 NPC1 (0.46) RAB9AKDRKITFLT3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed