SCHEMBL8090855

SCHEMBL8090855

O=C(c1cccc2ccccc12)N1CC(CN2CCC(CCCc3ccccc3)CC2)C(c2ccccc2)C1

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.75
CACNA1F O60840 2/20 0.58
CACNA1D Q01668 2/20 0.58
CACNA1S Q13698 2/20 0.58
CACNA1C Q13936 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7829388 0.90 CCR5 (0.79) CCR5
SCHEMBL7826171 0.87 CCR5 (0.70) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7839328 0.86 CCR5 (1.00) CCR5
SCHEMBL7829337 0.85 CCR5 (0.76) CCR5
SCHEMBL7983139 0.81 CCR5 (0.68) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7495984 0.81 CCR5 (0.68) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7833271 0.81 CCR5 (0.89) CCR5
SCHEMBL7832599 0.81 CCR5 (0.72) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7829234 0.80 CCR5 (0.60) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7838237 0.79 CCR5 (1.00) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166037-A Pyrrolidine and piperidine modulators of chemokine receptor activity MERCK & CO., INC. (US) 2000-12-26 US disclosed