SCHEMBL8091315

SCHEMBL8091315

NC(=O)Nc1ccc(CC[C@@H](O)CN2CCN(c3ccc(Cl)cc3)C2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.46
NPC1 O15118 1/20 0.42
CNR1 P21554 2/20 0.41
HDAC1 Q13547 8/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.38
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2023658 0.83 KCNH2 (0.68) KCNH2NPC1MAPT
SCHEMBL2023657 0.83 KCNH2 (0.68) KCNH2NPC1MAPT
SCHEMBL12576482 0.73 MAPT (0.68) KCNH2ADRB2ADRB1ADRB3MAPT
SCHEMBL14864581 0.72 MAPT (0.55) KCNH2MAPT
SCHEMBL2016782 0.67 KCNH2 (0.68) KCNH2ADRB2ADRB1ADRB3MAPT
SCHEMBL2016784 0.67 KCNH2 (0.68) KCNH2ADRB2ADRB1ADRB3MAPT
SCHEMBL2025770 0.66 KCNH2 (0.61) KCNH2DRD2DRD3MAPT
SCHEMBL2025768 0.66 KCNH2 (0.61) KCNH2DRD2DRD3MAPT
SCHEMBL12577213 0.65 TSHR (0.53) KCNH2MAPT
SCHEMBL430722 0.65 DRD2 (0.43) NPC1HDAC1DRD2DRD3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006437-A1 NMDA RECEPTOR ANTAGONISTS FOR NEUROPROTECTION EMORY UNIVERSITY (US) 2009-01-08 WO disclosed