SCHEMBL8091654

SCHEMBL8091654

CN(CCCCCc1ccccc1)C(C)(C)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.61
KCNH2 Q12809 3/20 0.49
AOC3 Q16853 1/20 0.47
FDPS P14324 3/20 0.46
TAAR1 Q96RJ0 1/20 0.44
GGPS1 O95749 1/20 0.43
CHRM2 P08172 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD1 P21728 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
ADRA1A P35348 1/20 0.43
OPRM1 P35372 1/20 0.43
DRD3 P35462 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8100038 0.98 SIGMAR1 (0.58) SIGMAR1KCNH2AOC3FDPSTAAR1
SCHEMBL8097390 0.93 AOC3 (0.55) SIGMAR1KCNH2AOC3FDPSTAAR1
SCHEMBL8084282 0.86 TAAR1 (0.55) SIGMAR1AOC3TAAR1
SCHEMBL9752620 0.83 KCNH2 (0.47) SIGMAR1KCNH2AOC3TAAR1CHRM2
SCHEMBL8099618 0.83 KCNH2 (0.47) SIGMAR1KCNH2AOC3CHRM2HTR1A
SCHEMBL8099117 0.77 SIGMAR1 (0.63) SIGMAR1
SCHEMBL8079373 0.76 SIGMAR1 (1.00) SIGMAR1KCNH2AOC3TAAR1
SCHEMBL9670745 0.76 SIGMAR1 (1.00) SIGMAR1KCNH2AOC3TAAR1
SCHEMBL2117266 0.76 SIGMAR1 (1.00) SIGMAR1KCNH2AOC3TAAR1
SCHEMBL22442307 0.76 SIGMAR1 (1.00) SIGMAR1KCNH2AOC3TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US claimed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP claimed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO claimed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO claimed