SCHEMBL8091784

SCHEMBL8091784

O=C(c1ccc(Cl)cc1)c1ccc(C=S)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.57
MAPK1 P28482 1/20 0.57
HPGD P15428 1/20 0.50
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
CYP1A2 P05177 1/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
MAOB P27338 2/20 0.44
CXCL12 P48061 1/20 0.44
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
NR4A1 P22736 1/20 0.44
MAOA P21397 1/20 0.43
ELANE P08246 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTT P42858 2/20 0.42
FABP2 P12104 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7506335 0.89 SRD5A2 (0.48) SRD5A2MAPK1HPGDHTTALDH1A1
SCHEMBL3081358 0.82
SCHEMBL1681512 0.82 SRD5A2 (0.80) SRD5A2MAPK1HPGDCES2CES1
SCHEMBL10697158 0.82 SRD5A2 (0.80) SRD5A2MAPK1HPGDCES2CES1
SCHEMBL9065412 0.82 SRD5A2 (0.80) SRD5A2MAPK1HPGDCES2CES1
SCHEMBL51827 0.82 SRD5A2 (0.80) SRD5A2MAPK1HPGDCES2CES1
SCHEMBL3565290 0.81 HSD17B10 (0.70) SRD5A2MAPK1HPGDCES2CES1
SCHEMBL4541125 0.81 ALDH1A1 (0.61) SRD5A2HPGDCES2CES1ALOX15
Hydrochloric Acid SCHEMBL11704986 0.79 SRD5A2 (0.76) SRD5A2MAPK1HPGDCES2CES1
SCHEMBL30010720 0.79 SRD5A2 (0.76) SRD5A2MAPK1HPGDCES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1058682-A1 HETEROCYCLIC DIARYLMETHYLENE DERIVATIVES, METHODS OF PREPARING THEM AND THEIR USES IN THERAPEUTICS LABORATOIRES UPSA (FR) 2000-12-13 EP disclosed
US-6004994-A ANTIINFLAMMATORY AGENTS, CYCLOOXYGENASE INHIBITORS AND ANALGESICS LABORATOIRES UPSA (FR) 1999-12-21 US disclosed
WO-1999043664-A1 HETEROCYCLIC DIARYLMETHYLENE DERIVATIVES, METHODS OF PREPARING THEM AND THEIR USES IN THERAPEUTICS LABORATOIRES UPSA (FR) 1999-09-02 WO disclosed