SCHEMBL8091889

SCHEMBL8091889

CCS(=O)(=O)Cc1cc(N)nc(-c2ccc(NC(=O)NCCCO)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.48
MTOR P42345 4/20 0.48
PIK3CD O00329 4/20 0.47
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 1/20 0.42
GLA P06280 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KDR P35968 4/20 0.41
PDGFRB P09619 1/20 0.41
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
HPGD P15428 1/20 0.38
APEX1 P27695 1/20 0.38
PTPN7 P35236 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8219107 0.92 PIK3CA (0.56) PIK3CAMTORPIK3CDKDM4ENPC1
SCHEMBL8098332 0.91 PIK3CA (0.48) PIK3CAMTORPIK3CDRAB9AKDR
SCHEMBL8098329 0.87 PIK3CA (0.55) PIK3CAMTORPIK3CDKDRPOLB
SCHEMBL8206121 0.85 PIK3CA (0.62) PIK3CAMTORPIK3CDKDM4ERAB9A
SCHEMBL8215045 0.85 PIK3CA (0.54) PIK3CAMTORPIK3CDKDRHDAC1
SCHEMBL11925678 0.84 PIK3CA (0.45) PIK3CAMTORPIK3CDKDM4ENPC1
SCHEMBL8215121 0.83 PIK3CA (0.56) PIK3CAMTORPIK3CDRAB9AKDR
SCHEMBL8213842 0.83 PIK3CA (0.57) PIK3CAMTORPIK3CDKDRPIK3CG
SCHEMBL8206190 0.83 PIK3CD (0.43) PIK3CAMTORPIK3CDKDM4EMEN1
SCHEMBL8084637 0.82 CA12 (0.45) PIK3CAMTORPIK3CDKDM4EHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed