SCHEMBL8092249

SCHEMBL8092249

C=CC[C@H](CN(C)C(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.53
TACR2 P21452 17/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099839 0.91 TACR1 (0.54) TACR1TACR2
SCHEMBL8582371 0.91 TACR1 (0.54) TACR1TACR2
SCHEMBL4258143 0.86 TACR1 (0.56) TACR1TACR2
SCHEMBL6594434 0.85 TACR1 (0.55) TACR1TACR2
SCHEMBL9110425 0.84 TACR2 (0.61) TACR1TACR2
SCHEMBL6598186 0.82 TACR1 (0.51) TACR1TACR2
SCHEMBL6424008 0.80 TACR2 (0.44) TACR1TACR2
SCHEMBL6424010 0.80 TACR2 (0.44) TACR1TACR2
SCHEMBL493651 0.80 TACR1 (0.48) TACR1
SCHEMBL3766497 0.80 TACR1 (0.48) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6013644-A AIDS THERAPY MERCK & CO., INC. (US) 2000-01-11 US disclosed
US-5869496-A TREATING ASTHMA, EMESIS MERCK & CO., INC. (US) 1999-02-09 US disclosed
EP-0681571-B1 SPIRO-SUBSTITUTED AZACYCLES AS TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1998-07-29 EP disclosed
WO-1998025604-A1 SPIRO-SUBSTITUTED AZACYCLES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1998-06-18 WO disclosed
EP-0681571-A1 SPIRO-SUBSTITUTED AZACYCLES AS TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 1995-11-15 EP disclosed
WO-1994017045-A1 SPIRO-SUBSTITUTED AZACYCLES AS TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1994-08-04 WO disclosed