SCHEMBL8092458

SCHEMBL8092458

Cc1cc(C)c(C)c(C(=O)Br)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38
ALDH1A1 P00352 3/20 0.36
TPMT P51580 1/20 0.34
METAP2 P50579 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
MYC P01106 1/20 0.33
ACHE P22303 1/20 0.33
LMNA P02545 1/20 0.33
CSNK2A1 P68400 1/20 0.33
NFE2L2 Q16236 1/20 0.33
DAO P14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1259080 0.79 KDM4E (0.47) KDM4ECA1CA2MMP1MMP2
SCHEMBL1259082 0.79 KDM4E (0.63) KDM4ECA1CA2MMP1MMP2
SCHEMBL13596324 0.79 KDM4E (0.47) KDM4ECA1CA2MMP1MMP2
SCHEMBL6910129 0.77 KDM4E (0.61) KDM4ECA1CA2MMP1MMP2
SCHEMBL6915538 0.77 KDM4E (0.61) KDM4ECA1CA2MMP1MMP2
SCHEMBL6914424 0.77 KDM4E (0.61) KDM4ECA1CA2MMP1MMP2
SCHEMBL6914098 0.77 KDM4E (0.61) KDM4ECA1CA2MMP1MMP2
SCHEMBL6915536 0.77 KDM4E (0.61) KDM4EALDH1A1TPMTMETAP2SMN1; SMN2
SCHEMBL6908359 0.77 KDM4E (0.61) KDM4ECA1CA2MMP1MMP2
SCHEMBL6916673 0.77 KDM4E (0.61) KDM4ECA1CA2MMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708077-B1 Diamino compounds and methods for preparing them CHISSO CORP (JP) 2000-12-27 EP disclosed
US-5663440-A Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1997-09-02 US disclosed
EP-0708077-A1 Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1996-04-24 EP disclosed