SCHEMBL8092545

SCHEMBL8092545

Cc1cc([N+](=O)[O-])c(C)cc1C(=O)Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
ALDH1A1 P00352 4/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
RECQL P46063 1/20 0.42
GPR35 Q9HC97 2/20 0.41
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
PDGFRB P09619 1/20 0.40
FGFR1 P11362 1/20 0.40
PDGFRA P16234 1/20 0.40
FLT1 P17948 1/20 0.40
FGFR3 P22607 1/20 0.40
KDR P35968 1/20 0.40
HSP90AA1 P07900 1/20 0.40
VCAM1 P19320 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11404100 0.93 TSHR (0.50) TSHRCES2CES1ALDH1A1CYP3A4
SCHEMBL773100 0.91 TSHR (0.47) TSHRCES2CES1ALDH1A1CYP1A2
SCHEMBL10627028 0.89 TSHR (0.46) TSHRCES2CES1ALDH1A1CYP1A2
SCHEMBL8142965 0.87 TSHR (0.43) TSHRCES2CES1ALDH1A1CYP1A2
SCHEMBL272650 0.83 TSHR (0.61) TSHRCES2CES1ALDH1A1CYP1A2
SCHEMBL1804737 0.83 TSHR (0.51) TSHRCES2CES1ALDH1A1CYP1A2
SCHEMBL10631279 0.82 TSHR (0.44) TSHRCES2CES1ALDH1A1CYP3A4
SCHEMBL8662780 0.82 TSHR (0.41) TSHRCES2CES1ALDH1A1GPR35
SCHEMBL8665268 0.82 TSHR (0.41) TSHRCES2CES1ALDH1A1GPR35
SCHEMBL8100252 0.81 TSHR (0.50) TSHRCES2CES1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708077-B1 Diamino compounds and methods for preparing them CHISSO CORP (JP) 2000-12-27 EP disclosed
US-5663440-A Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1997-09-02 US disclosed
EP-0708077-A1 Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1996-04-24 EP disclosed