SCHEMBL8100252

SCHEMBL8100252

Cc1cc([N+](=O)[O-])c(C)cc1C(=O)Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
CYP1A2 P05177 1/20 0.46
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
ALDH1A1 P00352 4/20 0.42
CYP3A4 P08684 1/20 0.42
RECQL P46063 1/20 0.42
GPR35 Q9HC97 2/20 0.41
MAPT P10636 4/20 0.40
RAB9A P51151 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
PDGFRB P09619 1/20 0.40
FGFR1 P11362 1/20 0.40
PDGFRA P16234 1/20 0.40
FLT1 P17948 1/20 0.40
FGFR3 P22607 1/20 0.40
KDR P35968 1/20 0.40
NPC1 O15118 2/20 0.40
GAA P10253 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL272650 0.83 TSHR (0.61) TSHRCYP1A2CES2CES1ALDH1A1
SCHEMBL1804737 0.83 TSHR (0.51) TSHRCYP1A2CES2CES1ALDH1A1
SCHEMBL8092545 0.81 TSHR (0.50) TSHRCYP1A2CES2CES1ALDH1A1
SCHEMBL1806976 0.81 TSHR (0.46) TSHRCYP1A2CES2CES1ALDH1A1
SCHEMBL8053279 0.79 TSHR (0.58) TSHRCYP1A2ALDH1A1CYP3A4RECQL
SCHEMBL273449 0.79 PDGFRB (0.62) TSHRCES2CES1ALDH1A1MAPT
SCHEMBL8136865 0.77 TSHR (0.58) TSHRCES2CES1ALDH1A1CYP3A4
SCHEMBL8129334 0.77 TSHR (0.58) TSHRCES2CES1ALDH1A1CYP3A4
SCHEMBL27862369 0.76 TSHR (0.72) TSHRCES2CES1ALDH1A1CYP3A4
SCHEMBL8094894 0.76 TSHR (0.72) TSHRALDH1A1MAPTRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708077-B1 Diamino compounds and methods for preparing them CHISSO CORP (JP) 2000-12-27 EP disclosed
US-5663440-A Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1997-09-02 US disclosed
EP-0708077-A1 Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1996-04-24 EP disclosed