SCHEMBL8092595

SCHEMBL8092595

C1CCC(CCCCCN2CCCCC2)CC1.c1ccc(CN2CCCCC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.58
SIGMAR1 Q99720 3/20 0.57
CCR3 P51677 1/20 0.54
ACHE P22303 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091980 0.89 SIGMAR1 (0.70) HRH3SIGMAR1CCR3
SCHEMBL4499239 0.82 CCR3 (0.69) SIGMAR1CCR3ACHE
SCHEMBL4499901 0.82 CCR3 (0.69) SIGMAR1CCR3ACHE
SCHEMBL7400077 0.82 SIGMAR1 (0.72) HRH3SIGMAR1CCR3
SCHEMBL7408920 0.82 SIGMAR1 (0.72) HRH3SIGMAR1CCR3
SCHEMBL9375727 0.82 HRH3 (0.62) HRH3SIGMAR1
SCHEMBL13978815 0.82 HRH3 (0.62) HRH3SIGMAR1
Hydrochloric Acid SCHEMBL7450136 0.81 SIGMAR1 (0.70) HRH3SIGMAR1CCR3
Hydrochloric Acid SCHEMBL7404498 0.81 SIGMAR1 (0.70) HRH3SIGMAR1CCR3
SCHEMBL12130736 0.80 HRH3 (0.58) HRH3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP disclosed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO disclosed