SCHEMBL8092937

SCHEMBL8092937

CCCCCN(Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1)c1c(N)cc[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 17/20 0.40
AGTR2 P50052 17/20 0.40
CXCR4 P61073 1/20 0.40
CMKLR1 Q99788 1/20 0.40
MAPK8 P45983 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092930 0.84 LTB4R2 (0.49) AGTR1
SCHEMBL8088498 0.77 MAPT (0.40)
SCHEMBL6844560 0.73 CXCR4 (0.42) AGTR1AGTR2CXCR4CMKLR1MAPK8
SCHEMBL8474830 0.73 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL9589057 0.73 AGTR1 (0.69) AGTR1AGTR2CXCR4CMKLR1MAPK8
SCHEMBL9590866 0.73 AGTR1 (0.71) AGTR1AGTR2
SCHEMBL8076371 0.73 AGTR1 (0.42) AGTR1AGTR2
SCHEMBL9295984 0.73 AGTR1 (0.45) AGTR1AGTR2CXCR4CMKLR1MAPK8
SCHEMBL9589717 0.73 AGTR1 (0.56) AGTR1AGTR2
SCHEMBL8088507 0.73 JAK2 (0.35) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6037349-A HAVING ANTAGONISTIC PROPERTIES TOWARDS ANGIOTENSIN II CAN BE USED FOR THE TREATMENT OF HYPERTENSION, ALDOSTERONISM AND CARDIAC INSUFFICIENCY MERCK PATENT GMBH (DE) 2000-03-14 US disclosed