SCHEMBL8092941

SCHEMBL8092941

CC(C)(C)OC(=O)N1CCC(Oc2ccc(CC(=O)N3CCC(N4C(=O)CCc5ccccc54)CC3)c(OCC(F)(F)F)c2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 14/20 0.67
AVPR2 P30518 6/20 0.67
AVPR1A P37288 6/20 0.67
HTR3E A5X5Y0 1/20 0.65
HTR3B O95264 1/20 0.65
CHRM4 P08173 1/20 0.65
HTR1A P08908 1/20 0.65
HTR1D P28221 1/20 0.65
HTR1B P28222 1/20 0.65
HTR2A P28223 1/20 0.65
HTR2C P28335 1/20 0.65
HTR1E P28566 1/20 0.65
HTR1F P30939 1/20 0.65
HTR7 P34969 1/20 0.65
ADRA1A P35348 1/20 0.65
DRD3 P35462 1/20 0.65
HTR2B P41595 1/20 0.65
HTR3A P46098 1/20 0.65
HTR5A P47898 1/20 0.65
HTR6 P50406 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357751 0.91 OXTR (0.77) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8089301 0.89 OXTR (0.85) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8089420 0.89 OXTR (0.81) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8081328 0.84 OXTR (0.76) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8089362 0.82 OXTR (0.69) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8081347 0.82 OXTR (0.75) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8081394 0.80 OXTR (1.00) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL8088568 0.80 OXTR (0.77) OXTRAVPR2AVPR1AHTR3EHTR3B
SCHEMBL7446609 0.80 OXTR (0.62) OXTRAVPR2AVPR1A
SCHEMBL7357703 0.80 OXTR (0.82) OXTRAVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed