SCHEMBL8092947

SCHEMBL8092947

c1ccc(CCCNC2CCCc3ccccc3C2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 1.00
GRIN2B Q13224 14/20 0.84
GRIN1 Q05586 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096625 0.91 GRIN2B (1.00) SIGMAR1GRIN2BGRIN1
SCHEMBL8092278 0.86 GRIN2B (1.00) SIGMAR1GRIN2BGRIN1
SCHEMBL8092549 0.83 GRIN2B (1.00) SIGMAR1GRIN2BGRIN1
SCHEMBL5142084 0.82 GRIN2B (0.82) SIGMAR1GRIN2B
SCHEMBL27929338 0.80 GRIN2B (0.71) SIGMAR1GRIN2BGRIN1
Hydrochloric Acid SCHEMBL9396249 0.79 GRIN2B (0.69) SIGMAR1GRIN2BGRIN1
SCHEMBL7325905 0.78 GRIN2B (0.70) SIGMAR1GRIN2BGRIN1
Hydrochloric Acid SCHEMBL7336883 0.77 GRIN2B (0.68) SIGMAR1GRIN2BGRIN1
Hydrochloric Acid SCHEMBL10447147 0.75 GRIN2B (0.96) SIGMAR1GRIN2BGRIN1
SCHEMBL388869 0.75 POLB (0.65) SIGMAR1GRIN2BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US claimed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP claimed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO claimed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO claimed