SCHEMBL8093648

SCHEMBL8093648

CC=C(CC)Oc1nc(-c2ccc(F)cc2)c(-c2ccc(S(C)(=O)=O)cc2)cc1C#N

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.54
PTGS1 P23219 4/20 0.54
CNR1 P21554 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8094098 0.91 PTGS2 (0.44) PTGS2PTGS1CNR1
SCHEMBL8098787 0.87 PTGS2 (0.52) PTGS2PTGS1CNR1
SCHEMBL8100740 0.85 PTGS2 (0.58) PTGS2PTGS1CNR1
SCHEMBL8098782 0.85 PTGS2 (0.54) PTGS2PTGS1CNR1
SCHEMBL8098785 0.85 PTGS2 (0.54) PTGS2PTGS1CNR1
SCHEMBL215205 0.84 PTGS2 (0.53) PTGS2PTGS1CNR1
SCHEMBL8092731 0.83 PTGS2 (0.64) PTGS2PTGS1CNR1
SCHEMBL8093419 0.82 PTGS2 (0.72) PTGS2PTGS1CNR1
SCHEMBL8093645 0.82 PTGS2 (0.53) PTGS2PTGS1CNR1
SCHEMBL8085292 0.82 PTGS2 (0.52) PTGS2PTGS1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP claimed
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed