SCHEMBL8093708

SCHEMBL8093708

CCCCOc1nc(-c2cccc(SC)c2)c(-c2ccc(S(N)(=O)=O)cc2)cc1CO

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.59
PTGS1 P23219 6/20 0.59
CA1 P00915 5/20 0.40
CA2 P00918 5/20 0.40
CA9 Q16790 5/20 0.40
CA7 P43166 2/20 0.40
CA12 O43570 2/20 0.40
TSHR P16473 1/20 0.40
CNR1 P21554 1/20 0.38
CA14 Q9ULX7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085593 0.92 PTGS2 (0.71) PTGS2PTGS1CNR1
SCHEMBL8095136 0.91 PTGS2 (0.66) PTGS2PTGS1CA1CA2CA9
SCHEMBL8094676 0.89 PTGS2 (0.61) PTGS2PTGS1CA1CA2CA9
SCHEMBL8094362 0.87 PTGS2 (0.59) PTGS2PTGS1CA1CA2CA9
SCHEMBL8094646 0.85 PTGS2 (0.42) PTGS2PTGS1CA1CA2CA9
SCHEMBL8085997 0.84 PTGS2 (0.68) PTGS2PTGS1CA1CA2CA9
SCHEMBL8776828 0.84 PTGS2 (0.67) PTGS2PTGS1CA1CA2CA9
SCHEMBL8093078 0.84 PTGS2 (0.83) PTGS2PTGS1CA1CA2CA9
SCHEMBL8423494 0.83 PTGS2 (0.42) PTGS2PTGS1CA1CA2CA9
SCHEMBL8093063 0.82 PTGS2 (0.80) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP claimed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP claimed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO claimed
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed