SCHEMBL8093865

SCHEMBL8093865

CS(=O)(=O)c1ccc(-c2cc(C#N)c(OCc3ccc4ccccc4n3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 8/20 0.52
PTGS2 P35354 5/20 0.47
PTGS1 P23219 2/20 0.47
CNR1 P21554 6/20 0.46
HTR2B P41595 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8086786 0.86 CNR1 (0.64) PTGS2PTGS1CNR1
SCHEMBL8095103 0.84 CNR1 (0.61) PTGS2PTGS1CNR1
SCHEMBL8092688 0.83 MAPK13 (0.43) PDE10APTGS2PTGS1
SCHEMBL8100740 0.82 PTGS2 (0.58) PTGS2PTGS1CNR1
SCHEMBL8095114 0.81 PTGS2 (0.58) PTGS2PTGS1CNR1
SCHEMBL8101395 0.81 CNR1 (0.55) PTGS2PTGS1CNR1
SCHEMBL8086370 0.81 PTGS2 (0.68) PTGS2PTGS1CNR1
SCHEMBL8096151 0.81 PTGS2 (0.49) PTGS2PTGS1CNR1
SCHEMBL8095250 0.81 PTGS2 (0.49) PTGS2PTGS1CNR1
SCHEMBL8092731 0.81 PTGS2 (0.64) PTGS2PTGS1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed