SCHEMBL8094036

SCHEMBL8094036

COc1ccc(-c2nc(Cl)c(C#N)cc2-c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.48
PTGS1 P23219 4/20 0.48
CNR1 P21554 2/20 0.47
CNR2 P34972 1/20 0.47
NPSR1 Q6W5P4 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
PAX8 Q06710 1/20 0.46
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CA12 O43570 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5904231 0.89 CNR1 (0.56) CNR1CNR2NPSR1ALDH1A1HPGD
SCHEMBL8093184 0.87 CNR1 (0.52) PTGS2PTGS1CNR1CNR2NPSR1
SCHEMBL8087025 0.86 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8085631 0.81 CNR1 (0.52) CNR1CNR2NPSR1ALDH1A1HPGD
SCHEMBL8099081 0.78 CNR1 (0.45) PTGS2PTGS1CNR1CNR2KDM4E
SCHEMBL8096139 0.78 KDM4E (0.54) PTGS2PTGS1CNR1CNR2NPSR1
SCHEMBL8093454 0.78 PTGS2 (0.45) PTGS2PTGS1CNR1CNR2KDM4E
SCHEMBL8095490 0.78 CNR1 (0.51) PTGS2PTGS1CNR1NPSR1ALDH1A1
SCHEMBL8092663 0.78 CNR1 (0.46) PTGS2CNR1CNR2KDM4E
SCHEMBL8098819 0.78 PTGS2 (0.43) PTGS2PTGS1CNR1CNR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed