SCHEMBL8096630

SCHEMBL8096630

CN(CCCCCc1ccccc1)CCCc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 1.00
AOC3 Q16853 1/20 0.62
FDPS P14324 3/20 0.60
GGPS1 O95749 1/20 0.58
KCNH2 Q12809 1/20 0.58
SLC6A2 P23975 1/20 0.57
SLC6A4 P31645 1/20 0.57
SLC6A3 Q01959 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11133953 0.98 SIGMAR1 (0.96) SIGMAR1AOC3FDPSGGPS1KCNH2
SCHEMBL7371550 0.94 SIGMAR1 (1.00) SIGMAR1FDPSGGPS1KCNH2
SCHEMBL12902332 0.94 SIGMAR1 (0.88) SIGMAR1AOC3FDPSKCNH2SLC6A2
SCHEMBL11134428 0.92 SIGMAR1 (0.96) SIGMAR1AOC3FDPSGGPS1SLC6A2
SCHEMBL29107028 0.90 SIGMAR1 (0.82) SIGMAR1AOC3KCNH2SLC6A2SLC6A4
SCHEMBL11131202 0.90 SIGMAR1 (0.82) SIGMAR1AOC3KCNH2SLC6A2SLC6A4
SCHEMBL19253990 0.90 SIGMAR1 (0.86) SIGMAR1FDPSGGPS1KCNH2
SCHEMBL8092655 0.90 SIGMAR1 (1.00) SIGMAR1FDPSGGPS1KCNH2SLC6A2
SCHEMBL11130673 0.90 SIGMAR1 (0.86) SIGMAR1FDPSGGPS1KCNH2
SCHEMBL11567562 0.90 SIGMAR1 (0.86) SIGMAR1FDPSGGPS1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US claimed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP claimed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO claimed
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP disclosed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO disclosed