SCHEMBL8097090

SCHEMBL8097090

Cc1cc(OC2CCN(Cc3ccccc3C(=N)NN=N)CC2)c2cccc(F)c2n1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.37
SCN1A P35498 4/20 0.36
SCN8A Q9UQD0 4/20 0.36
AR P10275 3/20 0.35
ACHE P22303 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
PHGDH O43175 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PDE4B Q07343 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091662 0.85 HRH1 (0.47) DRD4SCN1ASCN8AARKMT2A
SCHEMBL8095680 0.84 PDE4B (0.46) SCN1ASCN8AACHEOPRK1PHGDH
SCHEMBL13945410 0.79 MEN1 (0.39) DRD4ARMEN1KMT2A
SCHEMBL5526683 0.79 SCN1A (0.50) SCN1ASCN8A
SCHEMBL8088026 0.79 HTR2C (0.40) SCN1ASCN8AARACHEPDE4B
SCHEMBL8095861 0.79 KCNH2 (0.41) SCN1ASCN8AAR
SCHEMBL8102223 0.79 LMNA (0.40) DRD4MEN1KMT2A
SCHEMBL13968360 0.79 OPRL1 (0.42) DRD4AROPRL1MEN1KMT2A
SCHEMBL8094095 0.79 GRIN1 (0.40) SCN1ASCN8AARPHGDHMEN1
SCHEMBL8093682 0.77 SCN5A (0.40) SCN1ASCN8AARMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000085-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES USEFUL AS MODULATORS OF GATED ION CHANNELS PAINCEPTOR PHARMA CORPORATION (CA) 2008-12-31 WO disclosed