SCHEMBL8097537

SCHEMBL8097537

C[C@@H](n1ccn(-c2ccc(OCC(F)(F)C(F)F)cc2)c1=O)[C@@](O)(Cn1cncn1)c1ccccc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 14/20 0.42
CYP2C9 P11712 13/20 0.42
CYP2C19 P33261 13/20 0.42
CYP1A2 P05177 8/20 0.42
CYP2D6 P10635 8/20 0.42
KCNH2 Q12809 4/20 0.42
LMNA P02545 2/20 0.37
CYP2B6 P20813 1/20 0.37
CYP3A5 P20815 1/20 0.37
CYP3A7 P24462 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP3A43 Q9HB55 1/20 0.37
CYP46A1 Q9Y6A2 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8111206 1.00 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8105389 0.91 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8106906 0.91 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8097568 0.91 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8097483 0.91 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8669563 0.89 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9232324 0.89 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8538916 0.88 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8721176 0.87 CYP3A4 (0.50) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL7679956 0.85 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1033367-A2 Process for the preparation of optically active triazole derivatives and their imidazolidin-2-one intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-06 EP disclosed
US-5677464-A Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0687672-A2 Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-20 EP disclosed