SCHEMBL8097538

SCHEMBL8097538

C[C@@H](n1ccn(-c2ccc(OCC(F)(F)C(F)F)cc2)c1=O)[C@](O)(COS(C)(=O)=O)c1ccc(F)cc1F

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 10/20 0.34
CYP2C9 P11712 7/20 0.34
CYP2C19 P33261 7/20 0.34
CYP1A2 P05177 6/20 0.34
CYP2D6 P10635 6/20 0.34
KCNH2 Q12809 2/20 0.34
ACACB O00763 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
UGCG Q16739 1/20 0.30
KDM4E B2RXH2 1/20 0.30
TSHR P16473 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097541 1.00 CYP3A4 (0.34) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8097608 0.91 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8873890 0.91 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8106895 0.90 ACACB (0.32) KCNH2ACACBALDH1A1HTT
SCHEMBL8106891 0.90 ACACB (0.32) KCNH2ACACBALDH1A1HTT
SCHEMBL8105694 0.89 CYP3A4 (0.36) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8105698 0.89 CYP3A4 (0.36) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8111174 0.87 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8107346 0.87 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8105713 0.84 CYP3A4 (0.36) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1033367-A2 Process for the preparation of optically active triazole derivatives and their imidazolidin-2-one intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-06 EP disclosed
US-5677464-A Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0687672-A2 Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-20 EP disclosed