SCHEMBL8098767

SCHEMBL8098767

CSc1ccc(C2=CC[C@H]3[C@@H]4CC[C@H]5N(C)C(=O)CC[C@]5(C)[C@H]4CC[C@]23C)cc1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSD17B7 P56937 1/20 0.48
SRD5A1 P18405 1/20 0.47
SRD5A2 P31213 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084368 0.83 SRD5A1 (0.47) HSD17B7SRD5A1SRD5A2
SCHEMBL8083978 0.80 SRD5A1 (0.53) SRD5A1SRD5A2
SCHEMBL8952051 0.79 HSD17B7 (0.54) HSD17B7SRD5A1SRD5A2
SCHEMBL8952052 0.79 HSD17B7 (0.54) HSD17B7SRD5A1SRD5A2
SCHEMBL7524960 0.79 HSD17B7 (0.54) HSD17B7SRD5A1SRD5A2
SCHEMBL8951986 0.79 HSD17B7 (0.54) HSD17B7SRD5A1SRD5A2
SCHEMBL8951987 0.79 HSD17B7 (0.54) HSD17B7SRD5A1SRD5A2
SCHEMBL7524965 0.79 HSD17B7 (0.54) HSD17B7SRD5A1SRD5A2
SCHEMBL9211560 0.76 SRD5A1 (0.53) SRD5A1SRD5A2
SCHEMBL8072109 0.76 HSD17B7 (0.52) HSD17B7SRD5A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0756481-B1 17$g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO INC (US) 2000-12-27 EP disclosed
EP-0756481-A4 17-g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO INC (US) 1998-11-18 EP disclosed
EP-0756481-A1 17$g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO. INC. (US) 1997-02-05 EP disclosed
US-5525608-A ANTIACNE AGENT, SKIN DISORDERS, GLANDULAR DISORDERS MERCK & CO., INC. (US) 1996-06-11 US disclosed
WO-1995028928-A1 17β-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO., INC. (US) 1995-11-02 WO disclosed