SCHEMBL8098922

SCHEMBL8098922

COC(=O)C=C1CCCCCCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
HCAR2 Q8TDS4 2/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
ALDH1A1 P00352 3/20 0.33
HPGD P15428 3/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 4/20 0.33
HSD17B10 Q99714 2/20 0.33
ESR2 Q92731 1/20 0.32
SLC6A2 P23975 3/20 0.32
SLC6A3 Q01959 2/20 0.32
OPRK1 P41145 2/20 0.32
SLC6A4 P31645 1/20 0.32
SPR P35270 1/20 0.31
PRKCA P17252 2/20 0.31
CA12 O43570 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089816 1.00 TSHR (0.41) TSHRHCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL106091 1.00 TSHR (0.41) TSHRHCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL873013 0.98 TSHR (0.42) TSHRHCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL620969 0.93
SCHEMBL518574 0.88
SCHEMBL1187818 0.80 TSHR (0.43) TSHRHCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL1035256 0.80 TSHR (0.43) TSHRHCAR2KEAP1NFE2L2ALDH1A1
Hydrochloric Acid SCHEMBL23037273 0.78 TSHR (0.42) TSHRHCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL25223710 0.78 TSHR (0.46) TSHRHCAR2KEAP1NFE2L2ALDH1A1
SCHEMBL3264014 0.78 TSHR (0.39) TSHRHCAR2KEAP1NFE2L2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661271-B1 AZEPINE DERIVATIVES, PRODUCTION THEREOF, AND USE THEREOF AS SIGMA-RECEPTOR LIGANDS ASAHI CHEMICAL IND (JP) 2000-04-26 EP disclosed
US-5658923-A USED IN TREATING DISEASES RELATED TO SIGMA-RECEPTOR, SUCH AS SCHIZOPHRENIA ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1997-08-19 US disclosed
EP-0661271-A1 AZEPINE DERIVATIVE, PRODUCTION THEREOF, AND USE THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-07-05 EP disclosed