SCHEMBL8099277

SCHEMBL8099277

CC(=O)COc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.57
AKR1B1 P15121 1/20 0.57
ESR2 Q92731 1/20 0.51
PDCD1 Q15116 2/20 0.50
CD274 Q9NZQ7 2/20 0.50
PTPN1 P18031 1/20 0.47
PTPN5 P54829 1/20 0.45
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
S1PR1 P21453 1/20 0.44
S1PR3 Q99500 1/20 0.44
GRIA2 P42262 1/20 0.44
GRIA4 P48058 1/20 0.44
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
USP2 O75604 1/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8100940 0.86 FFAR1 (0.55) FFAR1AKR1B1ESR2PTPN1PTPN5
SCHEMBL8100769 0.84 FFAR1 (0.56) FFAR1AKR1B1ESR2PTPN1PTPN5
SCHEMBL8101456 0.81 NPC1 (0.53) FFAR1AKR1B1ESR2PTPN1PTPN5
SCHEMBL6960961 0.80 ESR2 (0.54) FFAR1AKR1B1ESR2PTPN1PTPN5
SCHEMBL6957583 0.79 ESR2 (0.56) FFAR1AKR1B1ESR2PTPN1PTPN5
SCHEMBL6959613 0.78 ESR2 (0.51) FFAR1AKR1B1ESR2PTPN1NPC1
SCHEMBL6961627 0.78 ESR2 (0.51) FFAR1AKR1B1ESR2PTPN1PTPN5
SCHEMBL7733929 0.76 MAPT (0.66) NPC1RAB9AALDH1A1HPGDUSP2
SCHEMBL3372818 0.76 MAPT (0.62) RAB9AALDH1A1HPGDMAPTCYP1A2
SCHEMBL30763519 0.76 ELANE (0.51) FFAR1AKR1B1ESR2PTPN1PTPN5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117885-A Biphenyl-substituted quinoline derivatives E. R. SQUIBB & SONS, INC. (US) 2000-09-12 US disclosed
EP-0556060-A1 Biphenyl-substituted quinoline and naphthyridines derivatives as angiotensine II antagonists E.R. SQUIBB & SONS, INC. (US) 1993-08-18 EP disclosed