SCHEMBL8100769

SCHEMBL8100769

CCCC(=O)COc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 3/20 0.56
AKR1B1 P15121 1/20 0.56
ALDH1A1 P00352 2/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
ESR2 Q92731 1/20 0.47
PTPN1 P18031 1/20 0.45
GRIA2 P42262 1/20 0.43
GRIA4 P48058 1/20 0.43
KDM4E B2RXH2 1/20 0.42
S1PR1 P21453 1/20 0.41
S1PR3 Q99500 1/20 0.41
PTPN5 P54829 1/20 0.41
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
HSD17B10 Q99714 2/20 0.41
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
MME P08473 1/20 0.40
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8100940 0.90 FFAR1 (0.55) FFAR1AKR1B1ALDH1A1HPGDTSHR
SCHEMBL8099277 0.84 FFAR1 (0.57) FFAR1AKR1B1ALDH1A1HPGDESR2
SCHEMBL6961627 0.79 ESR2 (0.51) FFAR1AKR1B1ALDH1A1HPGDTSHR
SCHEMBL6959613 0.79 ESR2 (0.51) FFAR1AKR1B1ALDH1A1HPGDESR2
SCHEMBL6960961 0.79 ESR2 (0.54) FFAR1AKR1B1ALDH1A1HPGDESR2
SCHEMBL8101456 0.77 NPC1 (0.53) FFAR1AKR1B1ALDH1A1ESR2PTPN1
SCHEMBL11573789 0.77 KDM4E (0.52) FFAR1AKR1B1ALDH1A1HPGDESR2
SCHEMBL9634048 0.76 KDM4E (0.54) FFAR1AKR1B1ALDH1A1HPGDTSHR
SCHEMBL4257509 0.76 KDM4E (0.54) FFAR1AKR1B1ALDH1A1HPGDTSHR
SCHEMBL6957583 0.74 ESR2 (0.56) FFAR1AKR1B1ALDH1A1HPGDESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117885-A Biphenyl-substituted quinoline derivatives E. R. SQUIBB & SONS, INC. (US) 2000-09-12 US disclosed
EP-0556060-A1 Biphenyl-substituted quinoline and naphthyridines derivatives as angiotensine II antagonists E.R. SQUIBB & SONS, INC. (US) 1993-08-18 EP disclosed