SCHEMBL8100686

SCHEMBL8100686

CS(=O)(=O)Nc1ccc(S(N)(=O)=O)cc1Nc1cccc(F)c1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 6/20 0.60
PTGS2 P35354 5/20 0.60
SOS1 Q07889 2/20 0.49
ALDH1A1 P00352 2/20 0.46
KMT2A Q03164 1/20 0.46
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA9 Q16790 3/20 0.44
CA12 O43570 2/20 0.44
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ESR1 P03372 1/20 0.43
PLA2G7 Q13093 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8105031 0.85 SOS1 (0.59) PTGS1PTGS2SOS1CA1CA2
SCHEMBL8092098 0.85 PTGS1 (0.60) PTGS1PTGS2ALDH1A1KMT2ACA1
SCHEMBL8105450 0.79 CA1 (0.47) PTGS2SOS1CA1CA2CA9
SCHEMBL8101123 0.77 PTGS1 (0.56) PTGS1PTGS2SOS1KMT2ACA1
SCHEMBL8099553 0.77 PTGS1 (0.56) PTGS1PTGS2SOS1CA1CA2
SCHEMBL8101694 0.76 CA2 (0.47) PTGS1PTGS2CA1CA2CA9
SCHEMBL8105340 0.75 PTGS1 (0.57) PTGS1PTGS2ALDH1A1KMT2ACA1
SCHEMBL8091420 0.74 CA2 (0.51) PTGS2SOS1CA1CA2CA9
SCHEMBL8091416 0.74 PTGS1 (0.56) PTGS1PTGS2KMT2ACA1CA2
SCHEMBL12811024 0.74 PTGS1 (0.57) PTGS1PTGS2ALDH1A1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed