SCHEMBL8101344

SCHEMBL8101344

CCCCOc1nc(-c2ccc(Br)cc2)c(-c2ccc(S(C)(=O)=O)cc2)cc1C#N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.58
PTGS1 P23219 5/20 0.58
CNR1 P21554 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.41
KDM4E B2RXH2 1/20 0.39
APAF1 O14727 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
PPARG P37231 1/20 0.39
KMT2A Q03164 1/20 0.39
NCOA2 Q15596 1/20 0.39
NCOA1 Q15788 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPK8 P45983 1/20 0.38
MAPK9 P45984 1/20 0.38
MAPK10 P53779 1/20 0.38
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8776763 0.92 PTGS2 (0.48) PTGS2PTGS1CNR1SMN1; SMN2TP53
SCHEMBL8086011 0.91 PTGS2 (0.59) PTGS2PTGS1CNR1KDM4EALDH1A1
SCHEMBL8094773 0.90 PTGS2 (0.58) PTGS2PTGS1CNR1
SCHEMBL8093419 0.90 PTGS2 (0.72) PTGS2PTGS1CNR1
SCHEMBL8086268 0.89 PTGS2 (0.57) PTGS2PTGS1CNR1MAPK8MAPK9
SCHEMBL8086370 0.87 PTGS2 (0.68) PTGS2PTGS1CNR1
SCHEMBL8087151 0.86 PTGS2 (0.67) PTGS2PTGS1CNR1
SCHEMBL8095038 0.86 PTGS2 (0.56) PTGS2PTGS1CNR1SMN1; SMN2KDM4E
SCHEMBL8086716 0.85 PTGS2 (0.53) PTGS2PTGS1CNR1
SCHEMBL8085692 0.85 KDM4E (0.42) PTGS2PTGS1CNR1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed