SCHEMBL8101397

SCHEMBL8101397

CCCC(=O)NC[C@@H]1C[C@H]1c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.55
MTNR1B P49286 12/20 0.54
MTNR1A P48039 11/20 0.54
CNR1 P21554 1/20 0.53
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HTR2B P41595 3/20 0.44
HTR2A P28223 2/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101400 1.00 HTR2C (0.55) HTR2CMTNR1BMTNR1ACNR1CYP3A4
SCHEMBL8098501 0.85 MTNR1B (0.52) HTR2CMTNR1BMTNR1AHTR2BHTR2A
SCHEMBL8095379 0.85 MTNR1B (0.52) HTR2CMTNR1BMTNR1ACNR1HTR2B
SCHEMBL8095382 0.85 MTNR1B (0.52) HTR2CMTNR1BMTNR1ACNR1HTR2B
SCHEMBL8098503 0.85 MTNR1B (0.52) HTR2CMTNR1BMTNR1AHTR2BHTR2A
SCHEMBL8096202 0.84 HTR2C (0.51) HTR2CMTNR1BMTNR1ACNR1HTR2B
SCHEMBL8098235 0.84 MTNR1B (0.54) MTNR1BMTNR1ACYP3A4CYP2C19L3MBTL1
SCHEMBL8098232 0.84 MTNR1B (0.54) MTNR1BMTNR1ACYP3A4CYP2C19L3MBTL1
SCHEMBL8098179 0.84 MTNR1B (0.51) HTR2CMTNR1BMTNR1AL3MBTL1HTR2B
SCHEMBL8088845 0.84 MTNR1B (0.51) HTR2CMTNR1BMTNR1AHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747346-B1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL MYERS SQUIBB CO (US) 2000-02-16 EP disclosed
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed
EP-0747346-A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed