SCHEMBL8102059

SCHEMBL8102059

COc1cccc(C2CC2(C)C(N)=O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.53
RCOR1 Q9UKL0 1/20 0.53
SLC9A1 P19634 2/20 0.51
PARP1 P09874 1/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
GLA P06280 2/20 0.46
GAA P10253 2/20 0.46
HPGD P15428 2/20 0.46
HTR2C P28335 4/20 0.43
HTR2A P28223 2/20 0.43
HTR2B P41595 2/20 0.43
DDB1 Q16531 1/20 0.43
CRBN Q96SW2 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15542258 0.78 KDM1A (0.55) KDM1ASLC9A1MAPK1CYP2C19
SCHEMBL6623618 0.78 KDM1A (0.55) KDM1ASLC9A1MAPK1CYP2C19
SCHEMBL28829972 0.78 KDM1A (0.60) KDM1ARCOR1SLC9A1KDM4EGAA
SCHEMBL15541944 0.78 KDM1A (0.55) KDM1ASLC9A1MAPK1CYP2C19
SCHEMBL28885396 0.75 KDM1A (0.51) KDM1ARCOR1SLC9A1ALDH1A1KDM4E
SCHEMBL15766833 0.71 KDM1A (0.97) KDM1ARCOR1HTR2CHTR2AHTR2B
SCHEMBL30997748 0.71 SLC9A1 (0.73) SLC9A1PARP1ALDH1A1KDM4EGLA
SCHEMBL15766835 0.71 KDM1A (0.97) KDM1ARCOR1HTR2CHTR2AHTR2B
SCHEMBL15780125 0.71 KDM1A (0.97) KDM1ARCOR1HTR2CHTR2AHTR2B
SCHEMBL2227972 0.70 KDM1A (0.36) KDM1AALDH1A1DDB1CRBNMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747346-B1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL MYERS SQUIBB CO (US) 2000-02-16 EP disclosed
EP-0747346-A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed