SCHEMBL8102085

SCHEMBL8102085

CCCc1cc([N+](=O)[O-])ccc1C(=O)Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
TP53 P04637 1/20 0.43
TDP1 Q9NUW8 4/20 0.43
ALDH1A1 P00352 4/20 0.43
CYP3A4 P08684 2/20 0.43
ALOX15 P16050 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
KMT2A Q03164 1/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.41
MAPT P10636 3/20 0.40
POLB P06746 2/20 0.40
ALOX5 P09917 1/20 0.40
MAPK1 P28482 1/20 0.40
BCL9 O00512 1/20 0.40
CTNNB1 P35222 1/20 0.40
TSHR P16473 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 1/20 0.40
EIF4A1 P60842 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8087236 0.91 ALDH1A1 (0.50) HTTTP53TDP1ALDH1A1CYP3A4
SCHEMBL8094971 0.90 ALDH1A1 (0.49) HTTTP53TDP1ALDH1A1KMT2A
SCHEMBL8094463 0.89 POLB (0.47) HTTTP53TDP1ALDH1A1CYP3A4
SCHEMBL8102118 0.89 ALDH1A1 (0.48) TDP1ALDH1A1EIF4A1
SCHEMBL8094302 0.89 ALDH1A1 (0.48) TDP1ALDH1A1EIF4A1
SCHEMBL8094160 0.89 ALDH1A1 (0.48) TDP1ALDH1A1EIF4A1
SCHEMBL3387313 0.86 ALDH1A1 (0.55) HTTTP53TDP1ALDH1A1CYP3A4
SCHEMBL8102317 0.85 KMT2A (0.45) HTTTP53TDP1ALDH1A1CYP3A4
SCHEMBL6272138 0.85 KMT2A (0.56) HTTTP53TDP1ALDH1A1CYP3A4
SCHEMBL14220842 0.79 KDM4E (0.49) HTTTDP1ALDH1A1CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708077-B1 Diamino compounds and methods for preparing them CHISSO CORP (JP) 2000-12-27 EP disclosed
US-5663440-A Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1997-09-02 US disclosed
EP-0708077-A1 Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1996-04-24 EP disclosed