SCHEMBL8102440

SCHEMBL8102440

CCOC(=O)CN(CCC#N)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TSHR P16473 1/20 0.36
ALDH1A1 P00352 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 1/20 0.35
CASP1 P29466 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
MLYCD O95822 2/20 0.34
CA14 Q9ULX7 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
CTSS P25774 3/20 0.32
CTSL P07711 2/20 0.32
CTSB P07858 2/20 0.32
CTSD P07339 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19643491 0.93 MEN1 (0.39) MEN1KMT2ATSHRALDH1A1SMN1; SMN2
SCHEMBL16336838 0.87 MEN1 (0.39) MEN1KMT2ATSHRALDH1A1SMN1; SMN2
SCHEMBL16710495 0.85 TSHR (0.38) TSHRALDH1A1MAPTCA12CA1
SCHEMBL23765759 0.83 CA12 (0.39) TSHRALDH1A1SMN1; SMN2CA12CA1
SCHEMBL18758783 0.83 CA12 (0.43) ALDH1A1SMN1; SMN2CA12CA1CA2
SCHEMBL22278113 0.82 CA14 (0.39) MEN1KMT2AALDH1A1SMN1; SMN2MAPT
SCHEMBL1280292 0.82 SSTR4 (0.40) ALDH1A1SMN1; SMN2CA12CA1CA2
SCHEMBL15312506 0.82 SMN1; SMN2 (0.38) TSHRALDH1A1SMN1; SMN2CA12CA1
SCHEMBL4517916 0.82 TSHR (0.37) TSHRALDH1A1MAPTCASP1MLYCD
SCHEMBL8028479 0.82 MLYCD (0.44) MEN1KMT2ATSHRALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104072498-A Synthetic method for (R)-N-[5-(2-methoxy-2-phenylacetyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole-3-yl]-4-(4-methyl piperazine-1-yl)benzamide UNIV SHENYANG PHARMACEUTICAL 2014-10-01 CN claimed
CN-104072498-B (R) synthetic method of N [5 (2 methoxyl group 2 phenyl acetyl) 1,4,5,6 nafoxidines also [3,4 c] pyrazoles 3 base] 4 (4 methyl piperazine 1 base) Benzoylamide 沈阳药科大学 2016-12-28 CN disclosed
CN-104072498-A Synthetic method for (R)-N-[5-(2-methoxy-2-phenylacetyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole-3-yl]-4-(4-methyl piperazine-1-yl)benzamide UNIV SHENYANG PHARMACEUTICAL 2014-10-01 CN disclosed
EP-1000931-A1 Process for producing an N-alkoxycarbonyl-N-cyanoethyl amino acid alkyl ester TOKUYAMA CORPORATION (JP) 2000-05-17 EP disclosed