SCHEMBL8102530

SCHEMBL8102530

CN(C(=O)Cc1ccccc1N(NS(C)(=O)=O)NS(C)(=O)=O)[C@@H](CC1CCCN1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 17/20 0.50
OPRD1 P41143 9/20 0.47
OPRM1 P35372 8/20 0.47
CYP2D6 P10635 7/20 0.47
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5629970 0.79 OPRK1 (0.78) OPRK1OPRD1OPRM1CYP2D6CYP3A4
Hydrochloric Acid SCHEMBL7978518 0.71 OPRK1 (0.40) OPRK1OPRD1OPRM1CYP2D6CYP3A4
Hydrochloric Acid SCHEMBL7978516 0.71 OPRK1 (0.40) OPRK1OPRD1OPRM1CYP2D6CYP3A4
SCHEMBL6478912 0.69 OPRK1 (0.64) OPRK1OPRD1OPRM1CYP2D6CYP3A4
SCHEMBL8102521 0.68 OPRK1 (0.35) OPRK1OPRD1OPRM1CYP2D6CYP3A4
SCHEMBL5631920 0.64 OPRK1 (0.77) OPRK1OPRD1OPRM1CYP2D6CYP3A4
SCHEMBL20832991 0.64 CYP2D6 (0.56) CYP2D6TSHR
SCHEMBL20833013 0.64 CYP2D6 (0.56) CYP2D6TSHR
SCHEMBL22259900 0.64 CYP2D6 (0.56) CYP2D6TSHR
SCHEMBL8507267 0.64 CYP2D6 (0.56) CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028063-A ADMINISTERING COMPOUND WITH OPIOID ACTIVITY ADOLOR CORPORATION (US) 2000-02-22 US claimed