SCHEMBL8103470

SCHEMBL8103470

CCC(C)(C)c1ccccc1N=C=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
TRPA1 O75762 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP3 P42574 1/20 0.33
RAB9A P51151 1/20 0.33
ATM Q13315 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TAAR1 Q96RJ0 1/20 0.31
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11280548 0.84 CYP3A4 (0.44) CYP3A4GABRA1GABRB2TRPA1ALDH1A1
SCHEMBL11280549 0.82 CYP3A4 (0.40) CYP3A4GABRA1GABRB2
SCHEMBL6544263 0.81 CYP3A4 (0.52) CYP3A4GABRA1GABRB2TRPA1ALDH1A1
SCHEMBL31318368 0.81 CYP3A4 (0.52) CYP3A4GABRA1GABRB2TRPA1ATM
SCHEMBL58726 0.81 CYP3A4 (0.52) CYP3A4GABRA1GABRB2TRPA1ATM
SCHEMBL4736911 0.79 CYP3A4 (0.43) CYP3A4GABRA1GABRB2TRPA1ALDH1A1
SCHEMBL12197004 0.78 CYP3A4 (0.38) CYP3A4GABRA1GABRB2TRPA1ALDH1A1
SCHEMBL6704455 0.76 CYP3A4 (0.47) CYP3A4GABRA1GABRB2TRPA1ALDH1A1
SCHEMBL10600545 0.76 NPC1 (0.36) NPC1LMNAMAPK1CASP3RAB9A
SCHEMBL10959911 0.74 CYP3A4 (0.39) CYP3A4GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed