SCHEMBL8104433

SCHEMBL8104433

CS(=O)(=O)c1ccc(C2CCC(=O)C2=Cc2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
LMNA P02545 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PTGS2 P35354 6/20 0.41
PTGS1 P23219 4/20 0.41
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
AKR1C3 P42330 1/20 0.38
XDH P47989 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8119635 1.00 CYP1A2 (0.43) CYP1A2LMNACYP2D6MAPTCYP2C19
SCHEMBL3438466 0.76 ALDH1A1 (0.49) CYP1A2LMNACYP2D6MAPTCYP2C19
SCHEMBL3438464 0.76 ALDH1A1 (0.49) CYP1A2LMNACYP2D6MAPTCYP2C19
SCHEMBL9047443 0.70 CYP1A2 (0.50) CYP1A2LMNACYP2D6MAPTCYP2C19
SCHEMBL9047452 0.70 CYP1A2 (0.50) CYP1A2LMNACYP2D6MAPTCYP2C19
SCHEMBL14223874 0.70 CYP1A2 (0.50) CYP1A2LMNACYP2D6MAPTCYP2C19
SCHEMBL3438392 0.70 HTT (0.43) CYP1A2LMNACYP2D6MAPTCYP2C19
SCHEMBL6163432 0.69 CYP1A2 (0.49) CYP1A2LMNACYP2D6MAPTCYP2C19
SCHEMBL3438205 0.68 MAPT (0.48) CYP1A2LMNAMAPTNPSR1
SCHEMBL3438204 0.68 MAPT (0.48) CYP1A2LMNAMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971910-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS Merck Frosst Canada & Co. (CA) 2000-01-19 EP disclosed
WO-1998043966-A1 ALPHA-METHYLENE GAMMA LACTONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA & CO. (CA) 1998-10-08 WO disclosed